Anacetrapib (MK-0859)

  • Anacetrapib (MK-0859)
Catalog No.: 3029

Anacetrapib (MK0859) is a potent, selective, reversible rhCETP and mutant CETP(C13S) inhibitor with IC50 of 7.9 nM and 11.8 nM, increases HDL-C and decreases LDL-C, does not increase aldosterone or blood pressure. Phase 3.

Chemical Name: 2-Oxazolidinone, 5-[3,5-bis(trifluoromethyl)phenyl]-3-[[4'-fluoro-2'-methoxy-5'-(1-methylethyl)-4-(trifluoromethyl)[1,1'-biphenyl]-2-yl]methyl]-4-methyl-, (4S,5R)-

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Biological Activity:
Anacetrapib (MK0859) is a potent, selective, reversible rhCETP and mutant CETP(C13S) inhibitor with IC50 of 7.9 nM and 11.8 nM, increases HDL-C and decreases LDL-C, does not increase aldosterone or blood pressure. Phase 3.
Technical Data:
M.W. 637.51
Formula: C30H25F10NO3
Solubility: DMSO
Purity: 98%
Storage: -20℃
CAS No: 875446-37-0
References:
Niesor EJ, et al. J Lipid Res. 2010, 51(12), 3443-3454. Ranalletta M, et al. J Lipid Res. 2010, 51(9), 2739-2752. Tan EY, et al. Drug Metab Dispos. 2010, 38(3), 459-473.

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Tags: Inhibitors, Metabolism, CETP, Anacetrapib (MK-0859), 875446-37-0

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